发明名称 |
NOVEL METHOD FOR THE SYNTHESIS OF (2S, 3AS, 7AS)-PERHYDROINDOLE-2-CARBOXYLIC ACID AND THE ESTERS THEREOF AND APPLICATION TO THE SYNTHESIS OF PERINDOPRIL |
摘要 |
<p>The invention relates to a method for the synthesis of derivatives of formula (I), where R= H or an acid-protecting group. Of application to the synthesis of perindopril and the pharmaceutically-acceptable salts thereof.</p> |
申请公布号 |
WO2004083237(A1) |
申请公布日期 |
2004.09.30 |
申请号 |
WO2004FR00592 |
申请日期 |
2004.03.12 |
申请人 |
LES LABORATOIRES SERVIER;DUBUFFET, THIERRY;LECOUVE, JEAN-PIERRE |
发明人 |
DUBUFFET, THIERRY;LECOUVE, JEAN-PIERRE |
分类号 |
C07D209/42;C07D225/02;C07K5/06;(IPC1-7):C07K5/02 |
主分类号 |
C07D209/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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