发明名称 TETRAHYDROPYRAN COMPOUNDS AS TACHYKININ ANTAGONISTS
摘要 <p>The present invention relates to the compounds of the formula (I), wherein R&lt;1&gt;, R&lt;2&gt;, R&lt;3&gt;, R&lt;4&gt;, R&lt;5&gt;, R&lt;6&gt;, R&lt;7&gt;, R&lt;8&gt;, R&lt;9&gt; and W are as defined herein, and pharmaceutically acceptable salts thereof; the compounds are of particular use in the treatment or prevention of depression, anxiety, pain, inflammation, migraine, emesis or postherpetic neuralgia.</p>
申请公布号 WO2004078750(A1) 申请公布日期 2004.09.16
申请号 WO2004GB00918 申请日期 2004.03.04
申请人 MERCK SHARP & DOHME LIMITED;DIRAT, OLIVIER;ELLIOTT, JASON, MATTHEW;HUSCROFT, IAN, THOMAS;JELLEY, RICHARD, ALEXANDER;KULAGOWSKI, JANUSZ, JOZEF;RAUBO, PIOTR, ANTONI;SHAW, DUNCAN, EDWARD;STERNFELD, FRANCINE;SWAIN, CHRISTOPHER, JOHN 发明人 DIRAT, OLIVIER;ELLIOTT, JASON, MATTHEW;HUSCROFT, IAN, THOMAS;JELLEY, RICHARD, ALEXANDER;KULAGOWSKI, JANUSZ, JOZEF;RAUBO, PIOTR, ANTONI;SHAW, DUNCAN, EDWARD;STERNFELD, FRANCINE;SWAIN, CHRISTOPHER, JOHN
分类号 A61P25/00;A61P29/00;C07D405/04;C07D405/06;C07D407/12;C07D417/04;C07D491/10;C07D498/04;(IPC1-7):C07D405/04;A61K31/40;A61K31/54;A61K31/435;A61K31/41 主分类号 A61P25/00
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