发明名称 PROCESS FOR SYNTHESISING USEFUL INTERMEDIATES FOR THE PREPARATION OF alphanubeta3 RECEPTOR ANTAGONISTS
摘要 The present invention relates to the synthesis of intermediates for the preparation of compounds of formula (A): wherein n is 2 or 3 and various salt forms of these compounds. The compounds of formula (A) are useful as alphanubeta3 receptor antagonists.
申请公布号 WO2004078109(A2) 申请公布日期 2004.09.16
申请号 WO2004GB00927 申请日期 2004.03.04
申请人 MERCK SHARP & DOHME LIMITED;MERCK & CO. INC.;BISHOP, BRIAN, CHRISTOPHER;BRANDS, KAREL, MARIE, JOSEPH;COTTRELL, IAN, FRANK;COWDEN, CAMERON, JOHN;DAVIES, ANTONY, JOHN;KEEN, STEPHEN, PHILIP;LIEBERMAN, DAVID, ROSS;STEWART, GAVIN, WILLIAM 发明人 BISHOP, BRIAN, CHRISTOPHER;BRANDS, KAREL, MARIE, JOSEPH;COTTRELL, IAN, FRANK;COWDEN, CAMERON, JOHN;DAVIES, ANTONY, JOHN;KEEN, STEPHEN, PHILIP;LIEBERMAN, DAVID, ROSS;STEWART, GAVIN, WILLIAM
分类号 C07D239/34;C07D405/04;C07D471/04 主分类号 C07D239/34
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