发明名称 |
TAXANE MIT CARBONATEN IN C-4 |
摘要 |
The present invention concerns novel taxane derivatives, their use as antitumor agents, and pharmaceutical formulations.The invention claims compounds of formula I and the use of compounds of formula I or pharmaceutical salts thereof as oral drugs for the treatment of human or veterinary disease.in which:R is phenyl, isopropyl, or tert butyl;R<1 >is -C(O)R<z >in which R<z >is (CH3)3CO-, (CH3)3CCH2-, CH3(CH2)3O-, cyclobutyl-, cyclohexyloxy, or (2-furyl);R<2 >is CH3C(O)O-. |
申请公布号 |
DE60012988(D1) |
申请公布日期 |
2004.09.16 |
申请号 |
DE2000612988 |
申请日期 |
2000.11.16 |
申请人 |
BRISTOL-MYERS SQUIBB CO., PRINCETON |
发明人 |
KADOW, F.;MASTALERZ, HAROLD;XUE, MAY;HANSEL, STEVEN;ZOECKLER, EDSON;ROSE, C.;TARRANT, G. |
分类号 |
A61K31/335;A61K31/337;A61K31/341;A61P35/00;C07D305/14;C07D407/12;(IPC1-7):A61K31/337 |
主分类号 |
A61K31/335 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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