发明名称 |
11beta LONG-CHAIN SUBSTITUTED ESTRATRIENES, METHOD FOR THEIR PRODUCTION, PHARMACEUTICAL PREPARATIONS CONTAINING SAID 11beta LONG-CHAIN SUBSTITUTED ESTATRIENES, AND THEIR USE FOR PRODUCING MEDICAMENTS |
摘要 |
This invention describes a 11beta-long-chain-substituted estratriene of general formula (I), in which R<11 >is a long-chain radical that has a nitrogen atom and optionally a sulfur atom, which in addition can be functionalized in the terminal position with a perfluoroalkyl group or an optionally substituted arly radical. The compound can have antiestrogenic or tissue-selective estrogenic properties and be suitable for the production of pharmaceutical agents.
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申请公布号 |
US6790842(B1) |
申请公布日期 |
2004.09.14 |
申请号 |
US20020018429 |
申请日期 |
2002.05.07 |
申请人 |
SCHERING AKTIENGESELLSCHAFT |
发明人 |
BOHLMANN ROLF;HEINRICH NIKOLAUS;KROLL JORG;SAUER GERHARD;FRITZEMEIER KARL-HEINRICH;HEGELE-HARTUNG CHRISTA;HOFFMANN JENS;LICHTNER ROSEMARIE;ZORN LUDWIG |
分类号 |
A61K31/565;A61K31/58;A61P5/30;A61P5/32;A61P17/14;A61P35/00;C07J1/00;C07J41/00;C07J43/00;(IPC1-7):A61K31/58;A61K31/56 |
主分类号 |
A61K31/565 |
代理机构 |
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代理人 |
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地址 |
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