发明名称 AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS
摘要 Aminopyridine and aminopyrazine compounds of formula (1), compositions including these compounds, and methods of their use are provided. Preferred compounds of formula 1 have activity as protein kinase inhibitors, including as inhibitors of c-MET.
申请公布号 CA2517256(A1) 申请公布日期 2004.09.10
申请号 CA20042517256 申请日期 2004.02.26
申请人 SUGEN, INC. 发明人 BOTROUS, IRINY;JOHNSON, JOANNE;LIN, JASON(QISHEN);FUNK, LEE A.;CHU, JI YU;NAMBU, MITCHELL DAVID;MENG, JERRY JIALUN;NELSON, CHRISTOPHER G.;TRAN-DUBE, MICHELLE;HARRIS, G. DAVIS, JR.;SHEN, HONG;BHUMRALKAR, DILIP;CUI, JINGJONG JEAN;WALTER, ALLISON;JIA, LEI;KOLODZIEJ, STEPHEN A.;KUNG, PEI-PEI;ZHANG, FANG-JIE;HANAU, CATHLEEN ELIZABETH;PAIRISH, MASON ALAN;ZHANG, JENNIFER;LI, XIAOYUAN(SHARON)
分类号 A61K;A61K31/496;A61K31/4965;A61K31/497;C07D;C07D211/72;C07D213/73;C07D401/00;C07D401/12;C07D403/00;C07D405/00;C07D409/00;C07D411/00;C07D413/00;C07D413/12;C07D417/00;C07D419/00;(IPC1-7):A61K31/496 主分类号 A61K
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