发明名称 ACETYLENE DERIVATIVES HAVING MGLUR 5 ANTAGONISTIC ACTIVITY
摘要 The invention provides compounds of formula I wherein n, A, R, R', R'', R0, X and Y are as defined in the description, and their preparation. The compounds of formula I are useful as pharmaceuticals.
申请公布号 EP1453512(A1) 申请公布日期 2004.09.08
申请号 EP20020792867 申请日期 2002.12.03
申请人 NOVARTIS AG 发明人 GASPARINI, FABRIZIO;AUBERSON, YVES;OFNER, SILVIO;HART, TERANCE W.;ZIMMERMANN, KASPAR
分类号 C07D215/26;A61K31/32;A61K31/4035;A61K31/405;A61K31/4439;A61K31/4709;A61K31/497;A61K31/5377;A61P25/00;A61P25/04;A61P25/14;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P25/34;A61P25/36;A61P43/00;C07C231/12;C07C233/18;C07C269/06;C07C271/16;C07D209/08;C07D209/36;C07D209/38;C07D209/44;C07D215/20;C07D401/04;C07D401/06;C07D405/04;C07D405/06;C07D405/12;(IPC1-7):A61K31/470;A61K31/404;C07D209/32;C07C233/23;C07C271/24 主分类号 C07D215/26
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