发明名称 Citrate salt of 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof
摘要 The present invention is directed to the citrate salt of 5,8,14-triazatetracyclo[10.3.1.0<2,11>.0<4,9>]-hexadeca-2(11),3,5,7,9-pentaene:and pharmaceutical compositions thereof. The present invention is also directed to the various forms of the citrate salt, particularly its hydrate and its anhydrous/nearly anhydrous polymorph. The invention is also directed to processes for preparation of these citrate salt forms.
申请公布号 US6787549(B2) 申请公布日期 2004.09.07
申请号 US20020139449 申请日期 2002.05.06
申请人 PFIZER INC. 发明人 JOHNSON PHILLIP J.;ROSE PETER R.;WILLIAMS GLENN R.;WINT LEWIN T.
分类号 C07D487/08;A61K;A61K31/495;A61K31/529;A61P;A61P1/04;A61P3/04;A61P5/14;A61P9/06;A61P9/12;A61P17/00;A61P17/02;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/10;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P25/36;A61P27/00;A61P29/00;A61P31/18;A61P39/02;C07D;C07D221/00;C07D223/00;C07D471/08;(IPC1-7):C07D471/08;A61K31/499 主分类号 C07D487/08
代理机构 代理人
主权项
地址