发明名称 |
Compostos e composições como inibidores de catepsina |
摘要 |
"COMPOSTOS E COMPOSIçõES COMO INIBIDORES DE CATEPSINA". A presente invenção refere-se a novos inibidores de catepsina S seletivos, seus sais farmaceuticamente aceitáveis e N-óxidos, seus usos como agentes terapêuticos e os métodos para sua fabricação.
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申请公布号 |
BR0210912(A) |
申请公布日期 |
2004.08.31 |
申请号 |
BR20020010912 |
申请日期 |
2002.06.03 |
申请人 |
AXYS PHARMACEUTICALS, INC.;AVENTIS PHARMACEUTICALS INC. |
发明人 |
MICHAEL GRAUPE;JIAYAO LI;JOHN O. LINK;SHEILA ZIPFEL;ANDREAS P. TIMM;DAVID J. ALDOUS;SUKANTHINI THURAIRATNAM |
分类号 |
C07D295/18;A61K31/165;A61K31/277;A61K31/341;A61K31/351;A61K31/381;A61K31/397;A61K31/40;A61K31/423;A61K31/4245;A61K31/426;A61K31/427;A61K31/428;A61K31/437;A61K31/4453;A61K31/4468;A61K31/454;A61K31/495;A61K31/5375;A61K31/5377;A61K31/55;A61P1/02;A61P13/12;A61P19/02;A61P21/04;A61P29/00;A61P33/06;A61P35/00;A61P43/00;C07C233/31;C07C255/29;C07C255/44;C07C255/46;C07C271/12;C07C271/16;C07C271/22;C07C271/24;C07C317/44;C07C317/46;C07C317/48;C07D205/04;C07D207/08;C07D207/16;C07D211/66;C07D223/08;C07D223/12;C07D239/08;C07D263/56;C07D271/06;C07D271/10;C07D277/28;C07D277/64;C07D277/82;C07D295/185;C07D295/20;C07D295/205;C07D307/14;C07D309/14;C07D333/24;C07D413/12;C07D413/14;C07D417/12;C07D498/04;(IPC1-7):C07D317/46;A61K31/16;C07 |
主分类号 |
C07D295/18 |
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