发明名称 |
PROTEIN KINASE C INHIBITOR |
摘要 |
THIS INVENTION PROVIDES NOVEL BIS-INDOLYLMALEIMIDE MACROCYCLE DERIVATIVES OF THE FORMULA: AND SOLVATES THEREOF. THE INVENTION FURTHER PROVIDES THE PREPARATION, PHARMACEUTICAL FORMULATIONS AND THE METHODS OF USE FOR INHIBITING PROTEIN KINASE C IN MAMMALS.
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申请公布号 |
MY118068(A) |
申请公布日期 |
2004.08.30 |
申请号 |
MYPI9604799 |
申请日期 |
1996.11.19 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
GARY LOWELL ENGEL;NAGY ALPHONSE FARID;MARGARET MARY FAUL;MICHAEL ROBERT JIROUSEK;LORI ANN RICHARDSON;LEONARD LARRY WINNEROSKI JR. |
分类号 |
A61K31/395;A61K31/40;A61K31/407;A61K31/44;A61P3/08;A61P3/10;A61P43/00;C07D471/04;C07D498/22 |
主分类号 |
A61K31/395 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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