发明名称 11beta-HALOGEN-7alpha-SUBSTITUTED ESTRATRIENES, PROCESS FOR THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS THAT CONTAIN THESE 11beta-HALOGEN-7alpha-SUBSTITUTED ESTRATRIENES AS WELL AS THEIR USE FOR THE PRODUCTION OF PHARMACEUTICAL AGENTS
摘要 This invention describes the new 11beta-halogen-7alpha-substituted estratrienes of general formula Iin whichR<11 >is a fluorine or chlorine atom, and the other substituents have the meanings that are explained in more detail in the description.The compounds have antiestrogenic properties or tissue-selective estrogenic properties and are suitable for the production of pharmaceutical agents.
申请公布号 US6780855(B2) 申请公布日期 2004.08.24
申请号 US19990380413 申请日期 1999.12.02
申请人 SCHERING AKTIENGESELLSCHAFT 发明人 BOHLMANN ROLF;HEINRICH NIKOLAUS;HOFMEISTER HELMUT;KROLL JORG;KUNZER HERMANN;SAUER GERHARD;ZORN LUDWIG;FRITZEMEIER KARL-HEINRICH;LESSL MONIKA;LICHTNER ROSEMARIE;NISHINO YUKISHIGE;PARCZYK KARSTEN;SCHNEIDER MARTIN
分类号 A61K31/565;A61K31/58;A61P5/32;A61P43/00;C07J31/00;C07J41/00;C07J43/00;(IPC1-7):C07J1/00;C07J17/00 主分类号 A61K31/565
代理机构 代理人
主权项
地址