发明名称 |
11beta-HALOGEN-7alpha-SUBSTITUTED ESTRATRIENES, PROCESS FOR THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS THAT CONTAIN THESE 11beta-HALOGEN-7alpha-SUBSTITUTED ESTRATRIENES AS WELL AS THEIR USE FOR THE PRODUCTION OF PHARMACEUTICAL AGENTS |
摘要 |
This invention describes the new 11beta-halogen-7alpha-substituted estratrienes of general formula Iin whichR<11 >is a fluorine or chlorine atom, and the other substituents have the meanings that are explained in more detail in the description.The compounds have antiestrogenic properties or tissue-selective estrogenic properties and are suitable for the production of pharmaceutical agents.
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申请公布号 |
US6780855(B2) |
申请公布日期 |
2004.08.24 |
申请号 |
US19990380413 |
申请日期 |
1999.12.02 |
申请人 |
SCHERING AKTIENGESELLSCHAFT |
发明人 |
BOHLMANN ROLF;HEINRICH NIKOLAUS;HOFMEISTER HELMUT;KROLL JORG;KUNZER HERMANN;SAUER GERHARD;ZORN LUDWIG;FRITZEMEIER KARL-HEINRICH;LESSL MONIKA;LICHTNER ROSEMARIE;NISHINO YUKISHIGE;PARCZYK KARSTEN;SCHNEIDER MARTIN |
分类号 |
A61K31/565;A61K31/58;A61P5/32;A61P43/00;C07J31/00;C07J41/00;C07J43/00;(IPC1-7):C07J1/00;C07J17/00 |
主分类号 |
A61K31/565 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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