发明名称 AVERMECTIN B1 DERIVATIVES HAVING AN AMINOSULFONYLOXY SUBSTITUENT IN THE 4''-POSITION
摘要 A compound of formula (I) wherein the bond marked by formula (II) indicates either the S or the R isomer at the 4''-position; and wherein R<SUB>1 </SUB>is C<SUB>1</SUB>-C<SUB>12</SUB>alkyl, C<SUB>3</SUB>-C<SUB>8</SUB>cycloalkyl; or C<SUB>2</SUB>-C<SUB>12</SUB>alkenyl; R<SUB>2 </SUB>is, for example, hydrogen, unsubstituted or mono- to penta-substituted C<SUB>1</SUB>-C<SUB>12</SUB>alkyl or unsubstituted or mono- to penta-substituted C<SUB>2</SUB>-C<SUB>12</SUB>alkenyl; R<SUB>3 </SUB>is, for example, hydrogen, C<SUB>1</SUB>-C<SUB>12</SUB>alkyl, mono- to penta-substituted C<SUB>1</SUB>-C<SUB>12</SUB>alkyl, unsubstituted or mono- to penta-substituted C<SUB>3</SUB>-C<SUB>12</SUB>cycloalkyl, or unsubstituted or mono- to penta-substituted C<SUB>2</SUB>-C<SUB>12</SUB>alkenyl; and wherein the substituents of the alkyl, alkenyl, alkynyl, alkylene, alkenylene and cycloalkyl radicals defined under R<SUB>2 </SUB>and R<SUB>3 </SUB>are selected, for example, from the group consisting of OH, halogen, halo-C<SUB>1</SUB>-C<SUB>2</SUB>alkyl, CN, NO<SUB>2 </SUB>and C<SUB>2</SUB>-C<SUB>6</SUB>alkynyl; and, where applicable, E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for the preparation of and the use of those compounds, their isomers and tautomers; starting materials for the preparation of the compounds of formula (I); pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a method of controlling pests using those compositions are described.
申请公布号 KR20040068335(A) 申请公布日期 2004.07.30
申请号 KR20047009873 申请日期 2002.12.20
申请人 发明人
分类号 C07D493/22;A01N25/04;A01N25/08;A01N43/90;C07D493/10;C07H17/08;C07H19/01 主分类号 C07D493/22
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