发明名称 Process for the preparation of dinapsoline
摘要 <p>A process for preparing a compound of formula (I), wherein R1 and R2 each are hydrogen; A is CH2, CHOH or C=O; R is hydrogen or C1-4alkyl, C1-4alkoxy, hydroxy or halogen. Also disclosed is a compound of formula (I), wherein R1 and R2 each are hydroxy-protecting group; or R1 and R2 may be joined together to form -(CH2)n-; n is 1 to 3; A is CHOR1 or C=O; R is hydrogen or C1-4alkyl; and R4, R5 and R6 each are independently hydrogen, C1-4alkyl, C1- 4alkoxy, hydroxy or halogen.</p>
申请公布号 NZ524212(A) 申请公布日期 2004.07.30
申请号 NZ20010524212 申请日期 2001.08.10
申请人 PURDUE RESEARCH FOUNDATION 发明人 SIT, SING-YUEN;JACUTIN-PORTE, SWANEE E
分类号 A61K31/473;A61K31/4741;A61P25/00;A61P25/16;A61P43/00;C07D221/18;C07D491/056;C07D491/06;(IPC1-7):A61K31/473;C07D471/00 主分类号 A61K31/473
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