发明名称 |
Compounds having both alpha7 nicotinic agonist activity and 5HT3 antagonist activity for the treatment of CNS diseases |
摘要 |
The invention discloses compounds that are selective alpha7 nAChR agonists and 5-HT3 antagonists. The compounds are useful for treating many CNS diseases.
|
申请公布号 |
US2004147522(A1) |
申请公布日期 |
2004.07.29 |
申请号 |
US20030698227 |
申请日期 |
2003.10.31 |
申请人 |
WONG ERIK HO FONG;CORTES-BURGOS LUZ A.;ROGERS BRUCE NELSON;PIOTROWSKI DAVID W.;WALKER DANIEL PATRICK;JACOBSEN ERIC JON;ACKER BRAD A.;WISHKA DONN G. |
发明人 |
WONG ERIK HO FONG;CORTES-BURGOS LUZ A.;ROGERS BRUCE NELSON;PIOTROWSKI DAVID W.;WALKER DANIEL PATRICK;JACOBSEN ERIC JON;ACKER BRAD A.;WISHKA DONN G. |
分类号 |
C07D453/02;C07D487/08;C07D519/00;(IPC1-7):A61K31/498;A61K31/474;A61K31/46 |
主分类号 |
C07D453/02 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|