发明名称 Acyl derivatives of 5-(2-(4-(1,2 benzisothiazole-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2h-indol-2-one having neuroleptic activity
摘要 A process for preparing acyl derivatives as prodrugs of 5-(2-(4-(1,2 benzisothiazole-3-yl)-1-piperazinyl)ethyl-6-chloro-1,3-dihydro-2H-indol-2-one and pharmaceutically acceptable acid addition salts and methods of use as an antipsychotic.
申请公布号 US2004138232(A1) 申请公布日期 2004.07.15
申请号 US20030689773 申请日期 2003.10.21
申请人 PFIZER INC 发明人 COLON-CRUZ ROBERTO;NORRIS TIMOTHY
分类号 A61P25/18;C07D417/12;(IPC1-7):A61K31/496;C07D417/14 主分类号 A61P25/18
代理机构 代理人
主权项
地址