发明名称 |
Acyl derivatives of 5-(2-(4-(1,2 benzisothiazole-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2h-indol-2-one having neuroleptic activity |
摘要 |
A process for preparing acyl derivatives as prodrugs of 5-(2-(4-(1,2 benzisothiazole-3-yl)-1-piperazinyl)ethyl-6-chloro-1,3-dihydro-2H-indol-2-one and pharmaceutically acceptable acid addition salts and methods of use as an antipsychotic.
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申请公布号 |
US2004138232(A1) |
申请公布日期 |
2004.07.15 |
申请号 |
US20030689773 |
申请日期 |
2003.10.21 |
申请人 |
PFIZER INC |
发明人 |
COLON-CRUZ ROBERTO;NORRIS TIMOTHY |
分类号 |
A61P25/18;C07D417/12;(IPC1-7):A61K31/496;C07D417/14 |
主分类号 |
A61P25/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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