发明名称 4(SPIROPIPERIDINYL)METHYL SUBSTITUTED PYRROLIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY
摘要 <p>3-Substituted pyrrolidines having a spiropiperidinylmethyl substituent on the 4-position of the ring are useful as modulators of chemokine receptor activity. In particular, these compounds are useful as modulators of the chemokine receptors CCR-3 and/or CCR-5.</p>
申请公布号 WO2004058763(A1) 申请公布日期 2004.07.15
申请号 WO2003US40491 申请日期 2003.12.19
申请人 MERCK & CO., INC.;BAO, JIANMING;BERESIS, RICHARD;BERGER, RICHARD;COLLETTI, STEVEN, L.;MIAO, SHOUWU;PARSONS, WILLIAM, H.;RUPPRECHT, KATHLEEN, M.;JOHANSON, JILL, N.;KAYSER, FRANK;KOVACS, ERNEST, W. 发明人 BAO, JIANMING;BERESIS, RICHARD;BERGER, RICHARD;COLLETTI, STEVEN, L.;MIAO, SHOUWU;PARSONS, WILLIAM, H.;RUPPRECHT, KATHLEEN, M.;JOHANSON, JILL, N.;KAYSER, FRANK;KOVACS, ERNEST, W.
分类号 A61K31/4355;A61K31/438;C07D491/10;C07D491/20;(IPC1-7):C07D471/10;A61K31/435 主分类号 A61K31/4355
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