发明名称 Oxa(thia)zolidine derivative and anti-inflammatory drug
摘要 The present invention provides medicinal compositions characterized by containing as the active ingredient either a compound represented by a general formula (1) or a pharmaceutically acceptable composite thereof,[wherein X represents oxygen or sulfur; R1 represents hydrogen, C1-4 alkyl, etc.; R2 represents, e.g., phenyl optionally substituted by A1; R3 represents, e.g., hydrogen, C1-4 alkyl optionally substituted by A2, or a group represented by either one of the following formulae;R represents oxygen, sulfur, or a group represented by a formula (N-G)], in particular, inhibitors of phospholipase A(2) activity; use of the compositions; and compounds represented by a general formula (1-1);wherein X, R1, R2, R3 and G1 are the same as defined in the description.
申请公布号 US6762200(B2) 申请公布日期 2004.07.13
申请号 US20020240075 申请日期 2002.09.25
申请人 NIPPON SODA CO. LTD. 发明人 TAKAGI MASAE;ISHIMITSU KEIICHI;NISHIBE TADAYUKI
分类号 A61K31/421;A61K31/422;A61K31/426;A61K31/427;A61K31/439;A61K31/4439;A61K31/454;A61K31/4709;A61K31/496;A61K31/506;A61K31/537;A61K31/5377;A61K31/54;A61P1/04;A61P1/16;A61P9/00;A61P9/02;A61P9/10;A61P11/00;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P25/00;A61P27/16;A61P29/00;A61P37/08;A61P43/00;C07D263/16;C07D263/26;C07D263/28;C07D277/14;C07D277/16;C07D277/18;C07D409/12;C07D413/04;C07D413/06;C07D413/10;C07D413/12;C07D417/04;C07D417/06;C07D417/12;C07D417/14;(IPC1-7):A61K31/44;C07D263/04 主分类号 A61K31/421
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