发明名称 |
COMPOSITIONS OF CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS AND HMG-COA REDUCTASE INHIBITORS |
摘要 |
A composition comprises (1) a solid amorphous adsorbate comprising a cholesteryl ester transfer protein (CETP) inhibitor and a substrate; and (2) an HMG-CoA reductase inhibitor. The solid amorphous adsorbate provides concentration enhancement of the CETP inhibitor relative to a control composition consisting essentially of the unadsorbed CETP inhibitor alone, resulting in improved bioavailability.
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申请公布号 |
CA2510458(A1) |
申请公布日期 |
2004.07.08 |
申请号 |
CA20032510458 |
申请日期 |
2003.12.18 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
BABCOCK, WALTER CHRISTIAN;SHANKER, RAVI MYSORE;SMITHEY, DANIEL TOD;FRIESEN, DWAYNE THOMAS |
分类号 |
A61K9/20;A61K31/40;A61K31/4706;A61K45/06;A61K45/08;A61P3/06;(IPC1-7):A61K45/06;A61K47/02;A61K47/32;A61K31/470 |
主分类号 |
A61K9/20 |
代理机构 |
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地址 |
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