发明名称 Compounds useful as reversible inhibitors of cysteine proteases
摘要 Disclosed are novel cathepsin S, K, F, L and B reversible inhibitory compounds of the formulas (I), (II), (Ia) and (Ib) further defined herein. The compounds are useful for treating autoimmune diseases. Also disclosed are processes for making such novel compounds.
申请公布号 US6756372(B2) 申请公布日期 2004.06.29
申请号 US20010001134 申请日期 2001.11.02
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 发明人 EMMANUEL MICHEL JOSE;LIU WEIMIN;SPERO DENICE MARY;SUN SANXING;THOMSON DAVID S.;WARD YANCEY DAVID
分类号 A61K31/40;A61K31/4468;A61K31/454;A61K31/496;A61K31/506;A61K31/517;A61K31/5365;A61K31/5377;A61K31/538;A61K31/541;A61K31/55;A61P1/04;A61P3/10;A61P9/10;A61P11/06;A61P19/10;A61P21/04;A61P25/28;A61P29/00;A61P31/00;A61P37/00;A61P37/06;C07D205/04;C07D207/14;C07D207/16;C07D211/58;C07D211/60;C07D211/66;C07D309/14;C07D335/02;C07D401/04;C07D401/12;C07D403/06;C07D405/12;C07D413/12;C07D413/14;C07D417/12;C07D455/02;C07D487/08;(IPC1-7):A61K31/535 主分类号 A61K31/40
代理机构 代理人
主权项
地址