| 发明名称 |
BENZOXAZIN-3-ONES AND DERIVATIVES THEREOF AS INHIBITORS OF PI3K |
| 摘要 |
<p>The present invention provides compounds of Formula (I) wherein W, Q, E, D, R<6>, R<7>, R<8>, Y, K, R<9>, R<1O>, R<12>, G, and the double bond denoted "*" have any of the values defined therefore in the specification, and pharmaceutically acceptable salts thereof, that are useful as agents in the treatment of diseases and conditions, including inflammatory diseases, cardiovascular diseases, and cancers. Also provided are pharmaceutical compositions comprising one or more compounds of Formula (I). The compounds are inhibitors of phosphoinsitide-3-kinase (P13K).</p> |
| 申请公布号 |
WO2004052373(A1) |
申请公布日期 |
2004.06.24 |
| 申请号 |
WO2003IB05451 |
申请日期 |
2003.11.25 |
| 申请人 |
WARNER-LAMBERT COMPANY LLC;BARVIAN, NICOLE, CHANTEL;KOLZ, CHRISTINE, NYLUND;PARA, KIMBERLY, SUZANNE;PATT, WILLIAM, CHESTER;VISNICK, MELEAN |
发明人 |
BARVIAN, NICOLE, CHANTEL;KOLZ, CHRISTINE, NYLUND;PARA, KIMBERLY, SUZANNE;PATT, WILLIAM, CHESTER;VISNICK, MELEAN |
| 分类号 |
C07D498/04;A61P29/00;A61K31/5513;A61K31/553;A61K31/554;C07D405/06;C07D413/06;C07D413/14;C07D417/06;C07D417/14;(IPC1-7):A61K31/538 |
主分类号 |
C07D498/04 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
|
| 地址 |
|
