EPOTHILONE ANALOGS FOR SITE SPECIFIC DELIVERY IN THE TREATMENT OF PROLIFERATIVE DISEASES
摘要
<p>Conjugates of epothilones and epothilone derivatives (as effectors) with suitable saccharides or saccharide derivatives (as recognition units) are described. Their production is carried out by the recognition units being reacted with suitable linkers, and the compounds that are produced are conjugated to the effectors. The pharmaceutical use of the conjugates for treating proliferative or angiogenesis-associated processes is described.</p>
申请公布号
WO2004050089(A1)
申请公布日期
2004.06.17
申请号
WO2003EP13780
申请日期
2003.12.05
申请人
SCHERING AG;BOSSLET, KLAUS;HESS-STUMPP, HOLGER;HOFFMANN, JENS;KLAR, ULRICH;ROTGERI, ANDREA
发明人
BOSSLET, KLAUS;HESS-STUMPP, HOLGER;HOFFMANN, JENS;KLAR, ULRICH;ROTGERI, ANDREA