发明名称 A PROCESS FOR THE PREPARATION OF 1-[[3-(6,7-DIHYDRO-1-METHYL-7-OXO-3-PROPYL-1H-PYRAZOLO[4,3-D]PYRIMIDINE-5-YL)-4-ETHOXYPHENYL]SULFONYL]-4-METHYLPIPERAZINE AND INTERMEDIARY COMPOUNDS
摘要 A process is provided for the preparation of a compound of formula (IA) (sidenafil/ViagraTM) comprising reacting a compound of formula (IIA) in the presence of -OR, wherein R in the case of formation of compound (IA) is cì2cì3 where X is a leaving group , (IA) (IIA).
申请公布号 UA66787(C2) 申请公布日期 2004.06.15
申请号 UA19990105491 申请日期 1999.10.08
申请人 PFIZER RESEARCH AND DEVELOPMENT COMPANY N.V./S.A. 发明人 DANN PETER JAMES;LEVETT PHILIPPE CHARLES
分类号 C07D295/22;A61K31/519;A61P15/10;C07D231/40;C07D231/54;C07D295/26;C07D401/02;C07D401/06;C07D487/00;C07D487/04;(IPC1-7):C07D487/04 主分类号 C07D295/22
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