发明名称 BORINIC ACID PROTEASE INHIBITORS
摘要 The invention provides compounds of formula I: wherein R<1>-R<4>, A, A<1>, and X have any the values described in the specification, as well as pharmaceutical compositions comprising such compounds, and methods of inhibiting proteases with such compounds. The invention also provides synthetic intermediates and processes useful for preparing compounds of formula (I).
申请公布号 WO03015706(A3) 申请公布日期 2004.06.03
申请号 WO2002US26300 申请日期 2002.08.16
申请人 WASHINGTON STATE UNIVERSITY RESEARCH FOUNDATION;YALE UNIVERSITY;MATTESON, DONALD, S.;FABRY-ASZTALOS, LEVENTE;PRUSOFF, WILLIAM, H.;PIVAZYAN, ARMAN, D. 发明人 MATTESON, DONALD, S.;FABRY-ASZTALOS, LEVENTE;PRUSOFF, WILLIAM, H.;PIVAZYAN, ARMAN, D.
分类号 A61K31/69;A61K38/00;C07F5/02;C07F7/18;C07K5/06;C07K5/08;C07K5/10 主分类号 A61K31/69
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