发明名称 |
IDOLE DERIVATIVES AS SOMATOSTATIN AGONISTS OR ANTAGONISTS |
摘要 |
The present invention provide a compound of the formula:wherein ring A represents an aromatic ring optionally having substituents; B, Y and Ya are the same or different and each represents a bond, etc.; R1 and R2 are the sa me or different and each represents a hydrogen atom, etc.; R3 represents a hydrogen atom, etc.; R4 and R5 are the same or different and each represents a hydrogen, etc.; R6 represents an indolyl group optionally having substituent s; and Z and Za are the same or different and each represents a hydrogen atom, etc.; or a salt thereof or a prodrug thereof, having a somatostatin receptor binding inhibition activity and is useful for preventing and/or treating diseases associated with somatostatin.
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申请公布号 |
CA2506735(A1) |
申请公布日期 |
2004.06.03 |
申请号 |
CA20032506735 |
申请日期 |
2003.11.18 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED |
发明人 |
MATSUNAGA, SHINICHIRO;TAKEKAWA, SHIRO;WATANABE, MASANORI;ABE, HIDENORI |
分类号 |
A61P3/04;A61P3/10;C07D209/20;C07D209/42;C07D401/12;C07D401/14;C07D403/12;C07D405/12;C07D405/14;C07D417/12;C07D417/14;C07D495/04;(IPC1-7):C07D209/20;A61K31/405;A61K31/454;A61K31/497 |
主分类号 |
A61P3/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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