发明名称 IDOLE DERIVATIVES AS SOMATOSTATIN AGONISTS OR ANTAGONISTS
摘要 The present invention provide a compound of the formula:wherein ring A represents an aromatic ring optionally having substituents; B, Y and Ya are the same or different and each represents a bond, etc.; R1 and R2 are the sa me or different and each represents a hydrogen atom, etc.; R3 represents a hydrogen atom, etc.; R4 and R5 are the same or different and each represents a hydrogen, etc.; R6 represents an indolyl group optionally having substituent s; and Z and Za are the same or different and each represents a hydrogen atom, etc.; or a salt thereof or a prodrug thereof, having a somatostatin receptor binding inhibition activity and is useful for preventing and/or treating diseases associated with somatostatin.
申请公布号 CA2506735(A1) 申请公布日期 2004.06.03
申请号 CA20032506735 申请日期 2003.11.18
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED 发明人 MATSUNAGA, SHINICHIRO;TAKEKAWA, SHIRO;WATANABE, MASANORI;ABE, HIDENORI
分类号 A61P3/04;A61P3/10;C07D209/20;C07D209/42;C07D401/12;C07D401/14;C07D403/12;C07D405/12;C07D405/14;C07D417/12;C07D417/14;C07D495/04;(IPC1-7):C07D209/20;A61K31/405;A61K31/454;A61K31/497 主分类号 A61P3/04
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