发明名称 |
4-hydroxy derivatives of 5,6,9,10-tetrahydro-10-((2-methyl-1h-imidazol-1-yl)methyl)-4h-pyrido-(3,2,1-jk)-carbazol-11(8h)-one |
摘要 |
The present invention relates to novel 4-hydroxy derivatives of 5,6,9,10-tetrahydro-10-Ä(2-methyl-1H-imidazol-1-yl)methylÜ-4H-pyrido-Ä3,2,1-jkÜ-carbazol-11(8H)-one with 5-HT3-receptor antagonistic activity. Furthermore, the invention relates to a process for the preparation of the novel derivatives.
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申请公布号 |
EP1424337(A1) |
申请公布日期 |
2004.06.02 |
申请号 |
EP20020026237 |
申请日期 |
2002.11.26 |
申请人 |
SOLVAY PHARMACEUTICALS GMBH |
发明人 |
BRUECKNER, REINHARD;EECKHOUT, CHRISTIAN;FINNER, EMIL;FRITSCH, HOLGER;RONKEN, ERIC;ROEST, MARCO;SANN, HOLGER;SCHMIDT, JOCHEN;VANDERMEIJ, PAUL |
分类号 |
A61P1/08;C07D401/06;(IPC1-7):C07D471/06;A61K31/437 |
主分类号 |
A61P1/08 |
代理机构 |
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地址 |
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