发明名称 2-Hydroxy-mutilin carbamate derivatives useful for antibacterial use
摘要 A 2-Hydroxy-mutilin carbamate derivative has the formula (I) wherein: R1 is a 5-or 6-membered optionally substituted heteroaryl group and R2 is vinyl or ethyl. The heteroaryl can be pyridine, pyridazine, pyrimidine, pyrazine, isoxazole, thiazole, imidazole, pyrazole, 1,2,3-triazole, 1,2,4-triazole, benzimidazole, 3-oxo-3,4-dihydropyrido[2,3-b] pyrazine, or pyrazolo[1,5-a] pyrimidine. The compounds are useful for treating microbial infections.
申请公布号 NZ521536(A) 申请公布日期 2004.05.28
申请号 NZ20010521536 申请日期 2001.03.29
申请人 SMITHKLINE BEECHAM P 发明人 BROOKS, GERALD;HUNT, ERIC;HOWARD, STEVEN
分类号 C07D237/24;A61K31/426;A61K31/44;A61K31/4409;A61K31/495;A61K31/4985;A61K31/50;A61K31/505;A61K31/519;A61P31/04;C07D213/81;C07D213/82;C07D233/61;C07D239/42;C07D241/26;C07D277/20;C07D277/56;C07D417/04;C07D471/04;C07D487/04;(IPC1-7):A61K31/44;A61K31/425;C07D231/16;C07D231/38;C07D239/34 主分类号 C07D237/24
代理机构 代理人
主权项
地址