发明名称 METHOD OF PREPARATION OF TERFENADINE AND ITS DERIVATIVES
摘要 <p>The invention relates to a new method of preparation of derivatives of piperidinyl butylphenylacetic acids. The compounds are histaminically active. The substances are prepared by Grignard reaction of alkylhalohydrins and suitably substituted aromatic aldehydes. The resulting diols are subjected to subsequent substitution reaction.</p>
申请公布号 WO2004043922(A1) 申请公布日期 2004.05.27
申请号 WO2003SK00021 申请日期 2003.11.07
申请人 ZENTIVA, A.S.;VEVERKA, MIROSLAV;BOHAC, ANDREJ;KRIZ, MIROSLAV;VARGA, IVAN 发明人 VEVERKA, MIROSLAV;BOHAC, ANDREJ;KRIZ, MIROSLAV;VARGA, IVAN
分类号 C07C33/26;C07C43/178;C07C69/732;C07D211/22;(IPC1-7):C07D211/22 主分类号 C07C33/26
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