发明名称 |
Acylated piperidine derivatives as melanocortin-4 receptor agonists |
摘要 |
Certain novel 4-substituted N-acylated piperidine derivatives are agonists of the human melanocortin receptor(s) and, in particular, are selective agonists of the human melanocortin-4 receptor (MC-4R). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the activation of MC-4R, such as obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.
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申请公布号 |
US2004097546(A1) |
申请公布日期 |
2004.05.20 |
申请号 |
US20030468515 |
申请日期 |
2003.08.19 |
申请人 |
GOULET MARK T.;NARGUND RAVI P.;SEBHAT IYASSU K.;UJJAINWALLA FEROZE;WALSH THOMAS F.;WARNER DANIEL;YE ZHIXIONG;YOUNG JONATHAN R.;BAKSHI RAMAN K. |
发明人 |
GOULET MARK T.;NARGUND RAVI P.;SEBHAT IYASSU K.;UJJAINWALLA FEROZE;WALSH THOMAS F.;WARNER DANIEL;YE ZHIXIONG;YOUNG JONATHAN R.;BAKSHI RAMAN K. |
分类号 |
A61K31/445;A61K31/451;A61K31/454;A61K31/4545;A61K31/5377;A61K45/00;A61P3/04;A61P3/10;A61P15/08;A61P15/10;A61P43/00;C07D211/62;C07D211/64;C07D401/04;C07D401/06;C07D401/14;C07D413/06;C07D413/14;C07D491/08;(IPC1-7):A61K31/454;C07D417/14;C0741/14 |
主分类号 |
A61K31/445 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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