ACYLOXYPYRROLIDINE DERIVATIVES AND USE THEREOF AS LIGANDS OF V1B OR BOTH V1B AND V1A RECEPTORS
摘要
The invention concerns acyloxypyrrolidine derivatives of general formula (I), wherein: R1 represents a hydrogen atom, a C1-C6 alkyl, a C3-C6 cycloalkyl, a -CH2CH2COOH group or a -NR2R3 group; R2 and R3 each independently represent a hydrogen atom or a C1-C6 alkyl. The invention also concerns a method for preparing said derivatives and their therapeutic use.
申请公布号
WO2004009585(A3)
申请公布日期
2004.05.06
申请号
WO2003FR02262
申请日期
2003.07.17
申请人
SANOFI-SYNTHELABO;AULOMBARD, ALAIN;GARCIA, GEORGES;PRADINES, ANTOINE;SERRADEIL-LE GAL, CLAUDINE;WAGNON, JEAN
发明人
AULOMBARD, ALAIN;GARCIA, GEORGES;PRADINES, ANTOINE;SERRADEIL-LE GAL, CLAUDINE;WAGNON, JEAN