发明名称 ACYLOXYPYRROLIDINE DERIVATIVES AND USE THEREOF AS LIGANDS OF V1B OR BOTH V1B AND V1A RECEPTORS
摘要 The invention concerns acyloxypyrrolidine derivatives of general formula (I), wherein: R1 represents a hydrogen atom, a C1-C6 alkyl, a C3-C6 cycloalkyl, a -CH2CH2COOH group or a -NR2R3 group; R2 and R3 each independently represent a hydrogen atom or a C1-C6 alkyl. The invention also concerns a method for preparing said derivatives and their therapeutic use.
申请公布号 WO2004009585(A3) 申请公布日期 2004.05.06
申请号 WO2003FR02262 申请日期 2003.07.17
申请人 SANOFI-SYNTHELABO;AULOMBARD, ALAIN;GARCIA, GEORGES;PRADINES, ANTOINE;SERRADEIL-LE GAL, CLAUDINE;WAGNON, JEAN 发明人 AULOMBARD, ALAIN;GARCIA, GEORGES;PRADINES, ANTOINE;SERRADEIL-LE GAL, CLAUDINE;WAGNON, JEAN
分类号 A61K31/404;A61P1/04;A61P3/04;A61P3/06;A61P3/10;A61P5/00;A61P9/00;A61P9/10;A61P13/12;A61P25/20;A61P25/22;A61P25/24;A61P35/00;C07D403/04 主分类号 A61K31/404
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