发明名称 Substituted carbazoles as inhibitors of spla2
摘要 Carbazoles of formula (I) with R<2>=hydroxyfunctional amide (hydroxamic or esters) are disclosed together with the use of such compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of conditions such as septic shock.
申请公布号 US2004087796(A1) 申请公布日期 2004.05.06
申请号 US20030467965 申请日期 2003.08.14
申请人 HARPER RICHARD WALTZ;LIN HO-SHEN;RICHETT MICHAEL ENRICO 发明人 HARPER RICHARD WALTZ;LIN HO-SHEN;RICHETT MICHAEL ENRICO
分类号 A61K31/403;A61P1/04;A61P1/18;A61P9/10;A61P11/00;A61P11/06;A61P19/00;A61P19/02;A61P19/06;A61P25/28;A61P27/14;A61P29/00;A61P31/00;A61P43/00;C07D209/88;C07D403/12;C07D409/04;(IPC1-7):C07D209/82;C0743/02 主分类号 A61K31/403
代理机构 代理人
主权项
地址