发明名称 |
Saccharin derivatives as orally active elastase inhibitors. |
摘要 |
Orally active compounds of general formula (I) wherein R1 is methyl, ethyl or 2-morpholino-ethyl group, R2 is piperidino, morpholino or 4-methyl-piperazinyl group, n is 2 or 3 and their salts, solvates and hydrates. |
申请公布号 |
ZA200204604(B) |
申请公布日期 |
2004.04.28 |
申请号 |
ZA20020004604 |
申请日期 |
2002.06.07 |
申请人 |
SANOFI-SYNTHELABO |
发明人 |
PETER ARANYI;STEPHANE DESSILLA;ZOLTAN KAPUI;ENDRE MIKUS;LAJOS T. NAGYI;KATALIN URBAN SZABO;LELLE VASVARINE DEBRECZY;SANDOR BATORI;ISTVAN HERMECZ;FERENC LEVAI;MARC PASCAL;BRUNO SIMONOT;MARTON VARGA |
分类号 |
A61K31/519;A61K31/5377;A61P1/04;A61P1/16;A61P1/18;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/10;A61P13/12;A61P17/00;A61P17/02;A61P17/06;A61P19/06;A61P25/00;A61P27/16;A61P29/00;A61P31/04;A61P31/10;A61P33/02;A61P33/12;A61P35/00;A61P37/02;A61P43/00;C07D471/04 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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