发明名称 CYCLOHEXYL SULPHONE DERIVATIVES AS GAMMA-SECRETASE INHIBITORS
摘要 Compounds of formula (I) inhibit the processing of APP by gamma-secretase, a nd hence are useful in treatment of Alzheimer's disease.
申请公布号 CA2500964(A1) 申请公布日期 2004.04.15
申请号 CA20032500964 申请日期 2003.09.25
申请人 MERCK SHARP & DOHME LIMITED 发明人 KERRAD, SONIA;OAKLEY, PAUL JOSEPH;WILLIAMS, SUSANNAH;HARRISON, TIMOTHY;CHURCHER, IAN;TEALL, MARTIN RICHARD;SHAW, DUNCAN EDWARD
分类号 C07C317/14;C07C317/18;C07C317/20;C07C317/22;C07C317/24;C07C317/44;C07C331/04;C07D205/04;C07D207/48;C07D211/96;C07D213/70;C07D213/71;C07D213/89;C07D233/84;C07D239/38;C07D249/08;C07D249/12;C07D257/04;C07D277/36;C07D285/12;C07D285/125;C07D295/092;C07D295/26;C07D307/38;C07D307/46;C07D307/52;C07D307/64;C07D307/68;C07D317/46;C07D333/18;C07D333/48;C07D491/08;(IPC1-7):C07C317/14;C07D205/06;C07D207/08;C07D295/08;C07D207/10;C07D207/16;C07D317/26;C07D211/38;C07D317/48 主分类号 C07C317/14
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