发明名称 Acetylenic alpha-amino acid-based sulfonamide hydroxamic acid tace inhibitors
摘要 Compounds of the formula:are useful in treating disease conditions mediated by TNF-alpha, such as rheumatoid arthritis, osteoarthritis, sepsis, AIDS, ulcerative colitis, multiple sclerosis, Crohn's disease and degenerative cartilage loss.
申请公布号 US6716833(B2) 申请公布日期 2004.04.06
申请号 US20030376871 申请日期 2003.02.27
申请人 WYETH HOLDINGS CORPORATION 发明人 LEVIN JEREMY I.;CHEN JAMES M.;COLE DEREK C.;DU MILA T.;LAAKSO LEIF M.
分类号 A61K31/5375;A61K31/54;C07C311/29;C07D213/68;C07D279/10;C07D279/12;C07D309/12;C07F9/36;(IPC1-7):A61K31/33;A61K31/18;C07D243/00;C07D223/00 主分类号 A61K31/5375
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