发明名称 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST
摘要 <p>A compound of the formula (I) wherein the variables X1 to X10, R&lt;1&gt; to R&lt;7&gt; including R&lt;3'&gt;, E, v, y, z, A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed.</p>
申请公布号 WO2004026305(A1) 申请公布日期 2004.04.01
申请号 WO2003US26300 申请日期 2003.09.17
申请人 ELI LILLY AND COMPANY;BLANCO-PILLADO, MARIA-JESUS;CHAPPELL, MARK, DONALD;DE LA TORRE, MARTA, GARCIA;DIAZ BUEZO, NURIA;FRITZ, JAMES, ERWIN;HOLLOWAY, WILLIAM, GLEN;MATT, JAMES, EDWARD, JUNIOR;MITCH, CHARLES, HOWARD;PEDREGAL-TERCERO, CONCEPCION;QUIMBY, STEVEN, JAMES;SIEGEL, MILES, GOODMAN;SMITH, DANA, RAE;STUCKY, RUSSELL, DEAN;TAKEUCHI, KUMIKO;THOMAS, ELIZABETH, MARIE;WOLFE, CHAD, NOLAN 发明人 DE LA TORRE, MARTA, GARCIA;BLANCO-PILLADO, MARIA-JESUS;CHAPPELL, MARK, DONALD;DIAZ BUEZO, NURIA;FRITZ, JAMES, ERWIN;HOLLOWAY, WILLIAM, GLEN;MATT, JAMES, EDWARD, JUNIOR;MITCH, CHARLES, HOWARD;PEDREGAL-TERCERO, CONCEPCION;QUIMBY, STEVEN, JAMES;SIEGEL, MILES, GOODMAN;SMITH, DANA, RAE;STUCKY, RUSSELL, DEAN;TAKEUCHI, KUMIKO;THOMAS, ELIZABETH, MARIE;WOLFE, CHAD, NOLAN
分类号 A61P3/04;C07C235/46;C07D213/38;C07D213/64;C07D213/643;C07D213/78;C07D213/81;C07D213/82;C07D217/04;C07D237/24;C07D241/24;C07D307/14;C07D333/20;C07D401/06;C07D401/12;C07D401/14;C07D405/12;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07D417/14;(IPC1-7):A61K31/441;A61K31/442;C07C43/20 主分类号 A61P3/04
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