发明名称 |
Spiro-indolines as Y5 receptor antagonists |
摘要 |
Compounds of general structural formula I such as that shown in structural formula II are selective NPY Y5 receptor antagonists, useful in the treatment of obesity and the complications associated therewith.
|
申请公布号 |
US2004063942(A1) |
申请公布日期 |
2004.04.01 |
申请号 |
US20030624414 |
申请日期 |
2003.07.21 |
申请人 |
MERCK & CO., INC.;BANYU PARMACEUTICAL CO., LTD. |
发明人 |
GAO YING-DUO;MACNEIL DOUGLAS J.;YANG LIHU;MORIN NANCY R.;FUKAMI TAKEHIRO;KANATANI AKIO;FUKURODA TAKAHIRO;ISHII YASUYUKI;IHARA MASAKI |
分类号 |
A61K31/403;A61K31/404;A61K31/4155;A61K31/4178;A61K31/4375;A61K31/438;A61K31/4427;A61K31/4439;A61K31/444;A61K31/4709;A61K31/497;A61K31/498;A61K31/501;A61K31/506;A61P3/04;A61P3/06;A61P3/10;A61P7/04;A61P9/04;A61P13/02;A61P15/00;A61P19/02;A61P25/04;A61P25/06;A61P25/08;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P37/02;C07D209/96;C07D221/20;C07D401/12;C07D403/12;C07D471/04;C07D471/10;C07D471/20;C07D487/10;C07D487/20;C07D519/00;(IPC1-7):C07D487/12;C07D471/12 |
主分类号 |
A61K31/403 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|