发明名称 CONDENSED BENZENE DERIVATIVE AND ITS USE
摘要 PROBLEM TO BE SOLVED: To provide a compound shown as general formula (I) useful for an androgen receptor modulator (especially agonist) having a non-steroid structure. SOLUTION: The compound or the salt is shown by general formula (I) and useful for an androgen receptor modulator. In the general formula, A ring is a (substituted) 5-membered or 8-membered hydrocarbon, B ring is a (substituted) 4-membered or 10-membered hydrocarbon, C ring is a (substituted) benzene ring, X<SP>1</SP>is carbon, X<SP>2</SP>is carbon, oxygen, etc., W is nitrogen, etc., Y<SP>11</SP>is shown as CR<SP>2</SP>R<SP>3</SP>' (R<SP>2</SP>is hydrogen, a cyano group, a nitro group, or the like, R<SP>3</SP>' is hydrogen, a cyano group, a nitro group, or the like), Y<SP>21</SP>is shown as CR<SP>4</SP>R<SP>5</SP>' (R<SP>4</SP>is hydrogen, a cyano group, a nitro group, or the like, R<SP>5</SP>' is hydrogen, a cyano group, a nitro group, or the like), and R<SP>1</SP>is an electron attractive group. Straight continuous-and-broken double line of the figure denotes a single bond or a double bond. COPYRIGHT: (C)2004,JPO
申请公布号 JP2004091486(A) 申请公布日期 2004.03.25
申请号 JP20030291584 申请日期 2003.08.11
申请人 TAKEDA CHEM IND LTD 发明人 SHIRAISHI MITSURU;HARA TAKAHITO;KUSAKA MASAMI;KANZAKI NAOYUKI;YAMAMOTO TETSUSHI;MIYAWAKI TOSHIO
分类号 C07D295/14;A61K31/045;A61K31/075;A61K31/122;A61K31/277;A61K31/336;A61K31/4015;A61K31/402;A61K31/4025;A61K31/4035;A61K31/415;A61K31/4152;A61K31/42;A61K31/438;A61K31/451;A61K31/4525;A61K31/4535;A61K31/472;A61K31/495;A61K31/535;A61K31/54;A61K31/55;A61K31/553;A61K45/00;A61P13/08;A61P15/12;A61P19/10;A61P35/00;A61P43/00;C07C255/53;C07C255/54;C07C255/56;C07D207/06;C07D207/08;C07D207/10;C07D207/12;C07D207/14;C07D207/16;C07D207/22;C07D207/24;C07D209/44;C07D211/14;C07D211/22;C07D211/28;C07D211/34;C07D211/42;C07D211/46;C07D211/60;C07D211/62;C07D211/74;C07D217/04;C07D231/22;C07D261/04;C07D265/02;C07D267/10;C07D303/46;C07D307/79;C07D409/04;C07D491/113;(IPC1-7):C07C255/53;A61K31/453;A61K31/452;A61K31/403;A61K31/401 主分类号 C07D295/14
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