发明名称 Imidazopyrimidine derivatives and triazolopyrimidine derivatives
摘要 A compound of the formula (I) wherein R<1 >is -X-R<4>, an optionally substituted heterocyclic residue, an optionally substituted carbocyclic residue or optionally substituted condensed ring moiety; X is CR<5>R<6>, O, S, SO, SO2 or NR<7>; Y is CH or N; R<2 >is H, an optionally substituted C1-C10 alkyl,etc.; R<3 >is an optionally substituted aryl, or an optionally substituted heteroaryl, etc.; R<4 >is an optionally substituted aryl, an optionally substituted heteroaryl, etc.; R<5>, R<6>, and R<7 >can be identical or different and represent H, an optionally substituted C1-C10 alkyl, etc. The compound has an excellent anti-allergic activity and the like.
申请公布号 US2004054179(A1) 申请公布日期 2004.03.18
申请号 US20030258628 申请日期 2003.02.14
申请人 YURA TAKESHI;CONCEPCION ARNEL B;HAN GYOONHEE;MARUMO MAKIKO;YOSHINO HIROKO;KAWAMURA NORIHIRO;KOKUBO TOSHIO;KOMURA HIROSHI;LI YINGFU;LOWINGER TIMOTHY B;MOGI MUNETO;YAMAMOTO NORIYUKI;YOSHIDA NAGAHIRO;MILLER SCOTT;POPP MARGARET A;REDMANN ANIKO M;RODRIGUEZ MARTHA E;SCOTT WILLIAM J;WANG MING 发明人 YURA TAKESHI;CONCEPCION ARNEL B;HAN GYOONHEE;MARUMO MAKIKO;YOSHINO HIROKO;KAWAMURA NORIHIRO;KOKUBO TOSHIO;KOMURA HIROSHI;LI YINGFU;LOWINGER TIMOTHY B;MOGI MUNETO;YAMAMOTO NORIYUKI;YOSHIDA NAGAHIRO;MILLER SCOTT;POPP MARGARET A;REDMANN ANIKO M;RODRIGUEZ MARTHA E;SCOTT WILLIAM J;WANG MING
分类号 A61K31/519;A61K31/5377;A61K31/541;A61P1/04;A61P3/04;A61P7/02;A61P7/06;A61P11/02;A61P11/06;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P21/04;A61P25/28;A61P27/02;A61P27/14;A61P29/00;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D487/04;C07D519/00;(IPC1-7):A61K31/519 主分类号 A61K31/519
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