发明名称 |
Thioaryl sulfonamide hydroxamic acid compounds |
摘要 |
A thioaryl sulfonamide hydroxamic acid compound that, inter alia, inhibits matrix metalloprotease activity is disclosed, as are a treatment process that comprises administering a contemplated thioaryl sulfonamide hydroxamic acid compound in a MMP enzyme-inhibiting effective amount to a host having a condition associated with pathological matrix metalloprotease activity.
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申请公布号 |
US2004034071(A1) |
申请公布日期 |
2004.02.19 |
申请号 |
US20030348419 |
申请日期 |
2003.01.21 |
申请人 |
GETMAN DANIEL P.;BECKER DANIEL P.;BARTA THOMAS E.;VILLAMIL CLARA I.;HOCKERMAN SUSAN L.;BEDELL LOUIS J.;LI MADELEINE HUI;FRESKOS JOHN N.;HEINTZ ROBERT M.;MC.DONALD JOSEPH J.;DECRESCENZO GARY A. |
发明人 |
GETMAN DANIEL P.;BECKER DANIEL P.;BARTA THOMAS E.;VILLAMIL CLARA I.;HOCKERMAN SUSAN L.;BEDELL LOUIS J.;LI MADELEINE HUI;FRESKOS JOHN N.;HEINTZ ROBERT M.;MC.DONALD JOSEPH J.;DECRESCENZO GARY A. |
分类号 |
C07D295/13;C07D309/12;(IPC1-7):C07D213/56;A61K31/44;A61K31/40;C07D207/08;C07C259/04 |
主分类号 |
C07D295/13 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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