Compounds, compositions and methods for modulating the activity of nuclear receptors are provided. In particular, heterocyclic compounds are provided for modulating the activity of farnesoid X receptor (FXR), liver X receptor (LXR) and/or orphan nuclear receptors. In certain embodiments, the compounds are thiazolidinone derivatives.
申请公布号
WO03060078(A9)
申请公布日期
2004.02.19
申请号
WO2002US41224
申请日期
2002.12.20
申请人
X-CEPTOR THERAPEUTICS, INC.;MARTIN, RICHARD;FLATT, BRENTON, TODD;WANG, TIE-LIN;KAHL, JEFFERY, DEAN
发明人
MARTIN, RICHARD;FLATT, BRENTON, TODD;WANG, TIE-LIN;KAHL, JEFFERY, DEAN