发明名称 |
NOVEL DRUGGABLE REGIONS IN SET DOMAIN PROTEINS AND METHODS OF USING THE SAME |
摘要 |
The present invention relates to novel druggable regions discovered in histo ne H3 lysine methyltransferase DIM-5, which is a SET domain protein. The presen t invention further relates to methods of using the druggable regions to scree n potential candidate therapeutics for diseases in which the activity of SET domain proteins are implicated, for example, anti-cancer/anti-proliferative agents or anti-fungal agents.
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申请公布号 |
CA2494837(A1) |
申请公布日期 |
2004.02.12 |
申请号 |
CA20032494837 |
申请日期 |
2003.08.06 |
申请人 |
EMORY UNIVERSITY |
发明人 |
XING, XHANG;XIAODONG, CHENG |
分类号 |
A61K;A61K6/00;A61K31/00;C12N9/10;C12N15/09;C12Q1/48;G01N23/20;G01N33/15;G01N33/50;G01N33/53;G01N33/573;G06F17/50;G06F19/16;(IPC1-7):C12N9/10;G06F19/00 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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