发明名称 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests.
摘要 Compounds of formula (I) and salts thereof:Wherein R<1 >represents methyl, ethyl, isopropyl or s-butyl; and R<2 >represents hydrogen or alkyl. R<3 >represents hydrogen, optionally substituted alkanoyl, optionally substituted alkenoyl, optionally substituted alkynoyl, alkylsulfonyl, or alkoxycarbonyl, or R<2 >and R<3 >together with the nitrogen atom to which they are attached form a saturated, optionally substituted 4- to 6-membered heterocyclic ring group. The moiety -a- together with the carbon atom to which it is attached forms a 3- to 6-membered cycloalkyl group. These compounds have anthelmintic, acaricidal and insecticidal activity.
申请公布号 ZA200208630(B) 申请公布日期 2004.02.12
申请号 ZA20020008630 申请日期 2002.10.24
申请人 SANKYO COMPANY, LIMITED 发明人 AKIO SAITO;TOSHIMITSU TOYAMA;YOKO SUGIYAMA;TOSHIHIKO NANBA
分类号 C07D493/22;A01N43/90;A01P5/00;A01P7/02;A01P7/04;C07H19/01 主分类号 C07D493/22
代理机构 代理人
主权项
地址