发明名称 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
摘要 Compounds of Formula (IA) and Formula (IB) wherein R<1>, R<2>, R<3>, R<4>, R<5>, and R<6 >are as defined herein for Formula (IA) or Formula (IB), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.
申请公布号 US2004023999(A1) 申请公布日期 2004.02.05
申请号 US20030394303 申请日期 2003.03.21
申请人 发明人 BEKKALI YOUNES;BETAGERI RAJASHEHAR;CARDOZO MARIO G.;GILMORE THOMAS A.;HARCKEN CHRISTIAN HANKE JUSTUS JOACHIM;KIRRANE THOMAS M.;KUZMICH DANIEL;PROUDFOOT JOHN ROBERT;RIETHER DORIS;TAKAHASHI HIDENORI;THOMSON DAVID S.;WANG JI;ZINDELL RENEE;RAZAVI HOSSEIN
分类号 A61K31/343;A61K31/404;A61K31/405;A61K31/4184;A61K31/423;A61K31/437;A61K31/44;A61K31/4402;A61K31/4439;A61P1/00;A61P1/16;A61P3/04;A61P3/10;A61P5/00;A61P9/00;A61P9/10;A61P9/12;A61P17/00;A61P19/02;A61P25/00;A61P25/04;A61P27/02;A61P27/06;A61P27/16;A61P29/00;A61P35/00;A61P37/06;A61P37/08;C07C49/255;C07C49/577;C07D209/12;C07D209/30;C07D213/30;C07D213/61;C07D215/14;C07D217/16;C07D231/12;C07D233/54;C07D235/12;C07D237/08;C07D239/26;C07D241/12;C07D261/18;C07D263/32;C07D263/56;C07D277/24;C07D277/64;C07D307/80;C07D333/16;C07D401/06;C07D405/06;C07D471/04;(IPC1-7):A61K31/513;A61K31/47;A61K31/428;A61K31/415;A61K31/381 主分类号 A61K31/343
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