发明名称 PHOSPHODIESTERASE 4 INHIBITORS, INCLUDING N-SUBSTITUTED ANILINE AND DIPHENYLAMINE ANALOGS
摘要 <p>PDE4 inhibition is achieved by novel compounds, e.g., N-substituted aniline and diphenylamine analogs. The compounds of the present invention are of Formula (I): wherein R&lt;1&gt;, R&lt;2&gt; R &lt;3&gt; and R&lt;4&gt; are as defined herein.</p>
申请公布号 WO2004009552(A1) 申请公布日期 2004.01.29
申请号 WO2003US22543 申请日期 2003.07.21
申请人 MEMORY PHARMACEUTICALS CORPORATION;SCHUMACHER, RICHARD, A.;HOPPER, ALLEN, T.;TEHIM, ASHOK;HESS, HANS-JURGEN, ERNST;UNTERBECK, AXEL;KUESTER, ERIK;BRUBAKER, WILLIAM, FREDERICK, JR.;DUNN, ROBERT, F. 发明人 SCHUMACHER, RICHARD, A.;HOPPER, ALLEN, T.;TEHIM, ASHOK;HESS, HANS-JURGEN, ERNST;UNTERBECK, AXEL;KUESTER, ERIK;BRUBAKER, WILLIAM, FREDERICK, JR.;DUNN, ROBERT, F.
分类号 A61K31/41;A61K31/135;A61K31/36;A61K31/40;A61K31/695;A61P25/00;C07C217/84;C07C217/86;C07C217/88;C07C217/92;C07C229/60;C07D213/38;C07D213/61;C07D213/68;C07D213/74;C07D213/75;C07D213/79;C07D213/80;C07D215/12;C07D215/14;C07D215/38;C07D217/22;C07D239/42;C07D241/12;C07D241/20;C07D261/08;C07D261/14;C07D277/28;C07D295/13;C07D307/14;C07D307/20;C07D317/58;C07D333/20;C07D401/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14;(IPC1-7):C07D213/38;C07D217/18;A61K31/44 主分类号 A61K31/41
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