发明名称 Rho-kinase inhibitors
摘要 Disclosed are compounds and derivatives thereof, their synthesis, and their use as Rho-kinase inhibitors. These compounds of the present invention are useful for inhibiting tumor growth, treating erectile dysfunction, and treating other indications mediated by Rho-kinase, e.g., coronary heart disease.
申请公布号 US2004014755(A1) 申请公布日期 2004.01.22
申请号 US20030339393 申请日期 2003.01.10
申请人 NAGARATHNAM DHANAPALAN;KHIRE UDAY;ASGARI DAVOUD;SHAO JIANXING;LIU XIAO-GAO;WANG CHUNGUANG;HART BARRY;WEBER OLAF;LYNCH MARK;ZHANG LEI;WANG LEI 发明人 NAGARATHNAM DHANAPALAN;KHIRE UDAY;ASGARI DAVOUD;SHAO JIANXING;LIU XIAO-GAO;WANG CHUNGUANG;HART BARRY;WEBER OLAF;LYNCH MARK;ZHANG LEI;WANG LEI
分类号 C07D491/048;A61K31/519;A61K31/5377;A61P7/02;A61P9/10;A61P9/12;A61P11/06;A61P15/10;A61P19/10;A61P25/00;A61P27/06;A61P35/00;A61P43/00;C07D471/04;C07D491/04;C07D495/04;(IPC1-7):A61K31/537;A61K31/517;C07D491/02;C07D498/02 主分类号 C07D491/048
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