PROCESS FOR THE SYNTHESIS OF HIV PROTEASE INHIBITORS
摘要
<p>An improved process for the synthesis of (3S)-tetrahydro-3-furyl N-[(1S,2R)-3 -(4-amino-N-isobutylbenzenesulphonamido)-1-benzyl-2-hydroxypropyl]carbamate comprising four steps form the compound of formula A and a novel intermediate thereto.</p>
申请公布号
HK1032047(A1)
申请公布日期
2004.01.09
申请号
HK20010102333
申请日期
2001.03.30
申请人
GLAXO GROUP LIMITED
发明人
AL-FARHAN, EMILE;DEININGER, DAVID D.;MCGHIE, STEPHEN;O'CALLAGHAN, JOHN;ROBERTSON, MARK STUART;RODGERS, KEITH;ROUT, STEPHEN JOHN;SINGH, HARDEV;TUNG, ROGER DENNIS