发明名称 |
2-(PHENYL)-2H-PYRAZOLE-3-CARBOXYLIC ACID-N-4-(THIOXO-HETEROCYCLYL)-PHENYL-AMIDE DERIVATIVES AND CORRESPONDING IMINO-HETEROCYCLYL DERIVATIVES AND RELATES COMPOUNDS FOR USE AS INHIBITORS OF THE COAGULATION FACTORS XA AND/OR VIIA FOR TREATING THROMBOSES |
摘要 |
The invention relates to the novel compounds of formula (I), wherein D, M, W , X, Y, T, R1 and R1~ are defined as in patent claim 1. The inventive compound s are inhibitors of coagulation factor Xa and can be used in the prophylaxis and/or therapy of thromboembolic diseases and in the treatment of tumors.</S DOAB>
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申请公布号 |
CA2491271(A1) |
申请公布日期 |
2004.01.08 |
申请号 |
CA20032491271 |
申请日期 |
2003.06.05 |
申请人 |
MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG |
发明人 |
GLEITZ, JOHANNES;BARNES, CHRISTOPHER;CEZANNE, BERTRAM;DORSCH, DIETER;MEDERSKI, WERNER;TSAKLAKIDIS, CHRISTOS |
分类号 |
A61K31/4155;A61K31/4178;A61K31/42;A61K31/433;A61P7/02;A61P9/08;A61P9/10;A61P25/06;A61P29/00;A61P35/00;A61P35/04;A61P43/00;C07D403/12;C07D413/14;C07D417/12;(IPC1-7):C07D417/14;C07D403/14;A61K31/415;A61K31/417;A61K31/422 |
主分类号 |
A61K31/4155 |
代理机构 |
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代理人 |
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地址 |
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