发明名称 THIAZOLE DERIVATIVES AS PHOSPHODIESTERASE IV INHIBITORS
摘要 The invention relates to thiazole derivatives of formula (I), in which R1, R 2, R3, V, W, X and B are defined as cited in claim 1. Said derivatives act as inhibitors of phosphodiesterase IV and can be used for treating osteoporosis , tumours, cachexia, arteriosclerosis, rheumatoid arthritis, multiple sclerosi s, diabetes mellitus, inflammatory processes, allergies, asthma, autoimmune diseases, myocardial diseases and AIDS.
申请公布号 CA2489902(A1) 申请公布日期 2003.12.31
申请号 CA20032489902 申请日期 2003.04.28
申请人 MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG 发明人 EGGENWEILER, HANS-MICHAEL;WOLF, MICHAEL
分类号 A61K31/501;A61P1/00;A61P1/04;A61P1/16;A61P3/10;A61P5/14;A61P7/00;A61P7/04;A61P7/06;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P11/08;A61P13/08;A61P13/12;A61P17/00;A61P17/02;A61P17/04;A61P17/06;A61P19/02;A61P19/06;A61P19/10;A61P21/04;A61P25/00;A61P25/14;A61P25/16;A61P25/24;A61P25/28;A61P27/02;A61P27/14;A61P29/00;A61P31/04;A61P31/10;A61P31/16;A61P31/18;A61P31/20;A61P31/22;A61P33/02;A61P33/06;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D417/06;C07D417/14;(IPC1-7):C07D417/14;A61K31/50 主分类号 A61K31/501
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