| 发明名称 |
CRYSTALLINE BISULPHATE SALT OF HIV PROTEASE AZAPEPTIDE INHIBITOR |
| 摘要 |
The invention relates to the crystalline bisulphate salt of the formula (I) which is found to have unexpectedly high solubility/dissolution rate and an oral bioavailability relative to the free base form of this HIV protease azapeptide inhibitor.
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| 申请公布号 |
RO118869(B1) |
申请公布日期 |
2003.12.30 |
| 申请号 |
RO20000000717 |
申请日期 |
1998.12.22 |
| 申请人 |
BRISTOL - MYERS SQUIBB COMPANY |
发明人 |
SINGH JANAK;PUDIPEDDI MADHUSUDHAN;LINDRUD MARK D. |
| 分类号 |
C07K5/02;A61K31/44;A61K31/4402;A61K31/4418;A61K38/05;A61P31/18;A61P43/00;C07D213/02;C07D213/42;(IPC1-7):C07D213/02 |
主分类号 |
C07K5/02 |
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