发明名称 SELECTIVE ENZYMATIC ESTERIFICATION AND SOLVOLYSIS OF EPIMERIC VITAMIN D ANALOG AND SEPARATION OF THE EPIMERS
摘要 Provided is a method of selectively enzymatically esterifying or selectively enzymatically solvolyzing epimers of analogs of vitamin D having a stereogenic center at C-24 that has a free or esterified OH group. The method can be used, for example, for separating mixed epimers of the vitamin D analog.
申请公布号 WO03060094(A3) 申请公布日期 2003.12.24
申请号 WO2003US00623 申请日期 2003.01.09
申请人 TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;SHAPIRO, EVGENY;FISHMAN, AYELET;EFFENBERGER, REINHARD;MAYMON, ASHER;SCHWARTZ, ANCHEL 发明人 SHAPIRO, EVGENY;FISHMAN, AYELET;EFFENBERGER, REINHARD;MAYMON, ASHER;SCHWARTZ, ANCHEL
分类号 C12P7/62;C12N9/20;C12P7/18;C12P41/00 主分类号 C12P7/62
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