发明名称 ASYMETRIC SYNTHESIS OF AMINO-PYRROLIDINONES
摘要 A novel process for the asymmetric synthesis of an amino-pyrrolidinone of the type shown below from appropriate pyrrolidinones is described. [Insert Chemical Formula] These compounds are useful as intermediates for MMP and TACE inhibitors.
申请公布号 WO03104220(A1) 申请公布日期 2003.12.18
申请号 WO2003US07969 申请日期 2003.03.14
申请人 BRISTOL-MYERS SQUIBB COMPANY;WALTERMIRE, ROBERT, E.;SAVAGE, SCOTT, A.;CAMPAGNA, SILVIO;MAGNUS, NICHOLAS, A.;CONFALONE, PASQUALE, N.;YATES, MATTHEW;MELONI, DAVID, J. 发明人 WALTERMIRE, ROBERT, E.;SAVAGE, SCOTT, A.;CAMPAGNA, SILVIO;MAGNUS, NICHOLAS, A.;CONFALONE, PASQUALE, N.;YATES, MATTHEW;MELONI, DAVID, J.
分类号 C07D207/26;C07D207/273;C07D401/12;(IPC1-7):C07D401/10;C07D207/04 主分类号 C07D207/26
代理机构 代理人
主权项
地址